1. Biopharmaceutics is concerned with the relationship between a drug's physicochemical properties, its dosage form, and the resulting therapeutic response after administration. 2. Factors like a drug's properties, dosage form characteristics, administration route and site of absorption influence the time course of the drug in plasma and its bioavailability. 3. Drug absorption can be influenced by physiological factors like membrane permeability, as well as physicochemical drug properties and dosage form design features.