Morphine and Related Drugs MedChem Ist Notes

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The document discusses several opioid drugs including morphine, codeine, meperidine, diphenoxylate, loperamide, fentanyl, methadone, propoxyphene, pentazocine, and levorphanol. It describes the mechanism of action and uses of each drug. The drugs derive analgesic effects through binding to opioid receptors in the brain and body and are used medically to treat pain or induce anesthesia. The document provides information on opioid drugs and their clinical applications.

Note
death
Morpheus
Ist

Introduction
raw opium
Uses of Morphine
10kg
1kg

Opioid Receptors
Naloxone Naltrexone
Ethylketazocine Bremazocine
DADLE DPDPE

MORPHINE DERIVATIVES
Naloxone Naltraxon nalorphine

Morphine and Its Structure
A
B C) D)
E

Morphine Sulphate
Mechanism of Action
Uses

Codeine
Mechanism of Action
Uses

Meperidine hydrochloride
Mechanism of Action
Uses:

Anilerdine hydrochloride
Mechanism of Action
Uses

Diphenoxylate Hydrochloride
Mechanism of Action
Uses

Loperamide Hydrochloride
Mechanism of Action
Uses:

Fentanyl citrate
Mechanism of Action
Uses

Methadone Hydrochloride
Mechanism of Action
Uses

Propoxyphene Hydrochloride
Mechanism of Action
Uses

Pentazocine
Mechanism of Action
Uses

LevorphanolTartrate
Mechanism of Action
6 to 8 times
Uses

Rahul Pal Mr. Abhishek Rai*
Saurabh Diwakar.

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