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ADRENERGIC
DRUG
TABLE OF CONTENTS:
Adrenergic Drugs?
What are Adrenergic Agonists? Sympathomimetic/ Adrenomimetics?
Types of stimulants?
What are adrenergic Antagonists/blockers?
Types of blockers?
Alpha-blockers Vs. Beta-blockers
References
Adrenergic Drugs:
Adrenergic drugs are medications that stimulate certain nerves in the body.
 by mimicking the action of the chemical messengers epinephrine and
norepinephrine
by stimulating their releases
Uses:
Uses in life threating conditions including : EXAMPLE: albuterol
` Salmeterol etc.
Cardiac arrest
Shock
Asthma attack
Allergic reaction
Adrenergic Agonists:
(Adrenomimetics)
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors.
Main Categories of Adrenergic receptors are:
Alpha (α1, α2 )→Anaphylactic shock, hypotension, nasal congestion and hemorrhage
Beta (β1, β2, and β3 ) → asthma, congestive heart failure.
Dopamine (D1-D5) → shock, congestive heart failure and Parkinson’s disease.
Drugs:
Isoproterenolum (β- adrenomimetic)
Fenoterolum (β2- adrenomimetic)
Dobutaminum (β1- adrenomimetic)
Terbutalinum
Galazolin(α-adrenomimetic)
Sympathomimetic Drugs:
Sympathomimetic drugs are stimulant compounds which mimic the
effects of agonists of the sympathetic nervous system.
Drugs: Catecholamine including:
I. Phenylephrine
II. Norepinephrine (noradrenaline)
III. Dopamine and epinephrine etc.
Uses of Drug(to treat):
Cardiac arrest
Hypotensive state
Allergic reaction
 Asthma etc.
Adrenergic antagonists
Adrenergic antagonists bind to the adrenoreceptors but do not trigger
the usual receptor-mediated intracellular effects.
Types :
• Alpha-blockers
• Beta-blockers
ALPHA-BLOCKERS Vs. BETA-
BLOCKERS
They relax certain muscles and help
small blood vessels remain open.
They work by keeping hormone
norepinephrine from tightening the
muscles in the walls of vessels which
causes them to remain relaxed. This
improves blood flow and lowers BP.
i.e;
Doxazosin and Prazoxin:
• Used to treat high BP
• Also used in men to treat enlarged
prostrate
Side effects:
• Might decrease low density
lipoprotein cholesterol (LDL)
They are also called blocking
agents, treat a variety of conditions
such as high BP and migraines.
Work by blocking the effects of
epinephrine. i.e;
Atenolol and Nadolol:
• Used to treat high blood pressure
• Migraines
• Can orally be taken and injections
also available
Side-effects:
• As same as a-blockers
Reference :
https://www.healthline.com/health/adrenergic-drugs
http://www.authorstream.com/Presentation/sachchidanand904-
1379392-sympathomimetic-drugs/
https://accessmedicine.mhmedical.com/content.aspx?bookid=1613&s
ectionid=102158209
https://www.kumc.edu/AMA-MSS/Study/pharm1_table.htm
ADRENERGIC DRUG

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ADRENERGIC DRUG

  • 2. TABLE OF CONTENTS: Adrenergic Drugs? What are Adrenergic Agonists? Sympathomimetic/ Adrenomimetics? Types of stimulants? What are adrenergic Antagonists/blockers? Types of blockers? Alpha-blockers Vs. Beta-blockers References
  • 3. Adrenergic Drugs: Adrenergic drugs are medications that stimulate certain nerves in the body.  by mimicking the action of the chemical messengers epinephrine and norepinephrine by stimulating their releases Uses: Uses in life threating conditions including : EXAMPLE: albuterol ` Salmeterol etc. Cardiac arrest Shock Asthma attack Allergic reaction
  • 4. Adrenergic Agonists: (Adrenomimetics) An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. Main Categories of Adrenergic receptors are: Alpha (α1, α2 )→Anaphylactic shock, hypotension, nasal congestion and hemorrhage Beta (β1, β2, and β3 ) → asthma, congestive heart failure. Dopamine (D1-D5) → shock, congestive heart failure and Parkinson’s disease. Drugs: Isoproterenolum (β- adrenomimetic) Fenoterolum (β2- adrenomimetic) Dobutaminum (β1- adrenomimetic) Terbutalinum Galazolin(α-adrenomimetic)
  • 5. Sympathomimetic Drugs: Sympathomimetic drugs are stimulant compounds which mimic the effects of agonists of the sympathetic nervous system. Drugs: Catecholamine including: I. Phenylephrine II. Norepinephrine (noradrenaline) III. Dopamine and epinephrine etc. Uses of Drug(to treat): Cardiac arrest Hypotensive state Allergic reaction  Asthma etc.
  • 6. Adrenergic antagonists Adrenergic antagonists bind to the adrenoreceptors but do not trigger the usual receptor-mediated intracellular effects. Types : • Alpha-blockers • Beta-blockers
  • 7. ALPHA-BLOCKERS Vs. BETA- BLOCKERS They relax certain muscles and help small blood vessels remain open. They work by keeping hormone norepinephrine from tightening the muscles in the walls of vessels which causes them to remain relaxed. This improves blood flow and lowers BP. i.e; Doxazosin and Prazoxin: • Used to treat high BP • Also used in men to treat enlarged prostrate Side effects: • Might decrease low density lipoprotein cholesterol (LDL) They are also called blocking agents, treat a variety of conditions such as high BP and migraines. Work by blocking the effects of epinephrine. i.e; Atenolol and Nadolol: • Used to treat high blood pressure • Migraines • Can orally be taken and injections also available Side-effects: • As same as a-blockers