1. Publication List
A. Papers
1. The acid mediated intramolecular 1,3- dipolar cycloaddition of 2- Nitro- 1,1
ethenediamine derived nitrile oxides for the synthesis of novel fused bicyclic
isoxazoles; Page, Lee W.;
Bailey, Matthew.; Beswick, Paul J.; Frydrych Simon.; Gleave, Robert J. for prospective
publication in Tetrahedron Letters (with the Editors)
2. The intramolecular amination of allenes; Feast, George C.; Page, Lee W.;
Robertson, Jeremy.; "in press" and can be cited as Chem. Commun., 2010, 46, DOI:10.1039/
b926179f
3. Synthesis and evaluation of 3- amino- 6- aryl- pyridazines as selective CB2
agonists for the treatment of inflammatory pain; Gleave, Robert J.; Beswick, Paul J.;
Brown, Andrew J.; Giblin, Gerard M. P.; Goldsmith, Paul; Haslam, Carl P.; Mitchell, William L.;
Nicholson, Neville H.; Page, Lee W.; Patel, Sadhana; Roomans, Susan; Slingsby, Brian P.;
Swarbrick, Martin E.; Bioorganic & Medicinal Chemistry Letters (2010), 20(2), 465-468.
CODEN: BMCLE8 ISSN:0960-894X. AN 2009:1591711 CAPLUS
4. An unusual methylene aziridine refined in P21/c and the nonstandard setting
P21/n; Feast, George C.; Haestier, James; Page, Lee W.; Robertson, Jeremy; Thompson,
Amber L.; Watkin, David J.; Acta Crystallographica, Section C: Crystal Structure
Communications (2009), C65(12), o635-o638. CODEN: ACSCEE ISSN:0108-2701. AN
2009:1534462 CAPLUS
5. 2- Amino- 5- aryl- pyridines as selective CB2 agonists: Synthesis and
investigation of structure- activity relationships. Gleave, Robert J.; Beswick, Paul J.;
Brown, Andrew J.; Giblin, Gerard M. P.; Haslam, Carl P.; Livermore, David; Moses, Andrew;
Nicholson, Neville H.; Page, Lee W.; Slingsby, Brian; Swarbrick, Martin E.; Bioorganic &
Medicinal Chemistry Letters (2009), 19(23), 6578-6581. CODEN: BMCLE8
ISSN:0960-894X. CAN 152:97308 AN 2009:1351270 CAPLUS
6. Identification of [4- [4- (methylsulfonyl)phenyl]- 6- (trifluoromethyl)- 2- pyrimidinyl]
amines and ethers as potent and selective cyclooxygenase- 2 inhibitors;
Swarbrick, Martin E.; Beswick, Paul J.; Gleave, Robert J.; Green, Richard H.; Bingham,
Sharon; Bountra, Chas; Carter, Malcolm C.; Chambers, Laura J.; Chessell, Iain P.; Clayton,
Nick M.; Collins, Sue D.; Corfield, John A.; Hartley, C. David; Kleanthous, Savvas; Lambeth,
Paul F.; Lucas, Fiona S.; Mathews, Neil; Naylor, Alan; Page, Lee W.; Payne, Jeremy J.;
Pegg, Neil A.; Price, Helen S.; Skidmore, John; Stevens, Alexander J.; Stocker, Richard;
Stratton, Sharon C.; Stuart, Alastair J.; Wiseman, Joanne O.; Bioorganic & Medicinal
Chemistry Letters (2009), 19(15), 4504-4508. CODEN: BMCLE8 ISSN:0960-894X. CAN
151:350051 AN 2009:845628 CAPLUS
B. Patents
1. Preparation of piperazine derivatives as cav2.2 calcium channel modulators;
Beswick, Paul John; Campbell, Alister; Cridland, Andrew Peter; Gleave, Robert James; Heer,
Jag Paul; Nicholson, Neville Hubert; Page, Lee William ; Vile, Sadie.; PCT Int. Appl.(2010),
65pp. CODEN: PIXXD2 WO 2010007072 A1 20100121 AN 2010:85019 CAPLUS
2. Preparation of piperazine derivatives as cav2.2 calcium channel modulators;
Beswick, Paul John; Campbell, Alister; Cridland, Andrew Peter; Gleave, Robert James; Heer,
Jag Paul; Nicholson, Neville Hubert; Page, Lee William ; Vile, Sadie.; PCT Int. Appl. (2010),
111pp. CODEN: PIXXD2 WO 2010007073 A1 20100121 AN 2010:85023 CAPLUS
3. Preparation of arylpyridazines as cannabinoid CB2 receptor agonists; Gleave,
Robert; Mitchell, William Leonard; Page, Lee William ; Swarbrick, Martin; Walters, Dewi
John.; PCT Int. Appl. (2007), 32pp. CODEN: PIXXD2 WO 2007022938 A2 20070301 CAN
146:274380 AN 2007:227874 CAPLUS.
4. Preparation of pyridazines as modulators of cannabinoid CB2 receptors; Gleave,
Robert; Mitchell, William Leonard; Page, Lee William ; Swarbrick, Martin.; PCT Int. Appl.
(2007), 44pp. CODEN: PIXXD2 WO 2007022937 A1 20070301 AN 2007:227298
CAPLUS.
5. Preparation of imidazopyridine derivatives as cannabinoid receptor ligands;
Eatherton, Andrew John; Giblin, Gerard Martin Paul; Mitchell, William Leonard; Naylor, Alan;
Page, Lee William ; Swarbrick, Martin; Sweeting, Jennifer Anne.; PCT Int. Appl. (2007),
58pp. CODEN: PIXXD2 WO 2007017237 A1 20070215 CAN 146:251845 AN
2007:173985 CAPLUS.