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DR.VIJAY NAGDEV H.O. MEDICAL UNIT-I CHANDKA MEDICAL COLLEGE LARKANA
Background ,[object Object],[object Object]
[object Object],[object Object]
MECHANISM OF ACTION ,[object Object],[object Object],[object Object]
Cont…. ,[object Object],[object Object]
RESISTANCE ,[object Object],[object Object],[object Object],[object Object]
[object Object]
Generations  Drugs  Spectrum  1 st (Quinolone) Nalidixic acid  Cinoxacin Gram-ve but not Pseudomonas species 2nd Norfloxacin Ciprofloxacin  Enoxacin  Ofloxacin  Gram- ve(including Pseudomonas species), some Gram+ (S. aureus) and some atypicals 3rd Levofloxacin  Sparfloxacin  Moxifloxacin Gemifloxacin Same as 2 nd  generation with extended Gram+ve and atypical coverage 4th *Trovafloxacin Same as 3 rd  generation with broad anaerobic coverage
Pharmacokinectics ,[object Object],[object Object],[object Object],[object Object],[object Object]
Distribution  ,[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
Drug interactions  Drugs increasing  levels of FQL FQL increasing the levels  of : Theophyline Antidepressants NSAIDS Imipramine  corticosteroids Caffene Theophyline Warfarin (INR –monitored)
 
 
Adverse effects. ,[object Object],[object Object],[object Object],[object Object],[object Object]
Cont. ,[object Object],[object Object],[object Object],[object Object]
Contraindication  ,[object Object],[object Object],[object Object],[object Object],[object Object]
[object Object]
Ciprofloxacin  ,[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
Clinical uses ,[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
[object Object],[object Object],[object Object],Oral  Parentral  Opthalmic  100 mg  200 mg iv 3mg/ml  solution 250 mg 400 mg iv 3.3mg/mg ointment 500 mg
Levofloxacin  ,[object Object],[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
Cont.  ,[object Object],[object Object],[object Object],[object Object],[object Object]
[object Object],[object Object],[object Object],Oral  Parentral  Opthalmic  100 mg  5 mg/ml iv 5mg/ml  solution 250 mg 25 mg/ml iv 500mg
 

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Fluoroquinolones

  • 1. DR.VIJAY NAGDEV H.O. MEDICAL UNIT-I CHANDKA MEDICAL COLLEGE LARKANA
  • 2.
  • 3.
  • 4.
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  • 6.
  • 7.
  • 8. Generations Drugs Spectrum 1 st (Quinolone) Nalidixic acid Cinoxacin Gram-ve but not Pseudomonas species 2nd Norfloxacin Ciprofloxacin Enoxacin Ofloxacin Gram- ve(including Pseudomonas species), some Gram+ (S. aureus) and some atypicals 3rd Levofloxacin Sparfloxacin Moxifloxacin Gemifloxacin Same as 2 nd generation with extended Gram+ve and atypical coverage 4th *Trovafloxacin Same as 3 rd generation with broad anaerobic coverage
  • 9.
  • 10.
  • 11. Drug interactions Drugs increasing levels of FQL FQL increasing the levels of : Theophyline Antidepressants NSAIDS Imipramine corticosteroids Caffene Theophyline Warfarin (INR –monitored)
  • 12.  
  • 13.  
  • 14.
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  • 20.
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  • 24. Â