Pharmacological
CLASSIFICATION OF DRUGS
with Doses and Preparations
FIFTH EDITION
KD Tripathi MD
Ex-Director-Professor and Head of Pharmacology
Maulana Azad Medical College and associated
LN and GB Pant Hospitals, New Delhi
JAYPEE BROTHERS MEDICAL PUBLISHERS (P) LTD
New Delhi • London • Philadelphia • Panama
®
1. Drugs Acting on Autonomic Nervous System .....................................................................................................................1
Cholinergic Drugs, Anticholinergic Drugs, Ganglionic Stimulants, Ganglionic Blocking Agents, Adrenergic Drugs,
-Adrenergic Blocking Drugs, -Adrenergic Blocking Drugs, Topical Drugs for Glaucoma
2. Autacoids and Related Drugs.................................................................................................................................................16
Histaminergic Agonists, H1-Antagonists, 5-Hydroxytryptamine (5-HT) Antagonists, Drugs for Migraine, Prostaglandins
(PGs), Nonsteroidal Antiinflammatory Drugs (NSAIDs)/Antipyretic Analgesics, Antirheumatoid Drugs, Drugs for Gout
3. Drugs for Respiratory Disorders............................................................................................................................................29
Drugs for Cough, Drugs for Bronchial Asthma
4. Hormones and Related Drugs ................................................................................................................................................37
Anterior Pituitary Hormones, Drugs Altering Anterior Pituitary Hormone Secretion, Thyroid Hormone, Thyroid Inhibitors,
Insulins, Oral Antidiabetic Drugs, Corticosteroids, Topical Steroids, Androgens and Related Drugs, Drugs for Erectile
Dysfunction, Estrogens and Related Drugs, Progestins, Hormonal Contraceptives, Uterine Stimulants, Uterine Relaxants
5. Drugs Acting on Peripheral (somatic) Nervous System...................................................................................................60
Skeletal Muscle Relaxants, Local Anaesthetics
6. Drugs Acting on Central Nervous System ..........................................................................................................................64
General Anaesthetics, Preanaesthetic Medication Drugs, Sedative-Hypnotic Drugs, Antiepileptic Drugs, Antiparkinsonian
Drugs, Antipsychotic Drugs, Drugs for Mania and Bipolar Disorder, Hallucinogens, Antidepressants, Antianxiety Drugs,
Opioid Analgesics and Antagonists, Central Nervous System (CNS) Stimulants, Cognition Enhancers
7. Cardiovascular Drugs ...............................................................................................................................................................88
Antihypertensive Drugs, Antianginal Drugs, Drugs for Peripheral Vascular Diseases, Drugs for Congestive Heart Failure,
Antiarrhythmic Drugs
Contents
Pharmacological Classification of Drugs with Doses and Preparations
xii
8. Drugs Acting on Kidney........................................................................................................................................................102
Diuretics, Antidiuretics
9. Drugs Affecting Blood ...........................................................................................................................................................105
Haematinics, Coagulants, Anticoagulants, Fibrinolytics, Antifibrinolytics, Antiplatelet Drugs, Hypolipidaemic Drugs,
Plasma Expanders
10. Gastrointestinal Drugs ...........................................................................................................................................................118
Drugs for Peptic Ulcer, Antiemetics, Laxatives, Drugs for Diarrhoea
11. Antibacterial Drugs.................................................................................................................................................................130
Antibacterial Drugs, Sulfonamides, Quinolone Antimicrobials, Penicillins, Cephalosporins, Monobactams, Carbapenems,
Aminoglycoside Antibiotics, Tetracyclines, Chloramphenicol, Macrolide Antibiotics, Lincosamide Antibiotics, Aminocyclitol
Antibiotic, Glycopeptide Antibiotics, Oxazolidinone, Polypeptide Antibiotics, Urinary Antiseptics, Antitubercular Drugs,
Antileprotic Drugs
12. Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs....................................................................................150
Antifungal Drugs, Antiviral Drugs (Non-retroviral), Antiretrovirus Drugs, Antimalarial Drugs, Antiamoebic Drugs,
Drugs for Giardiasis, Drugs for Trichomoniasis, Drugs for Leishmaniasis, Anthelmintic Drugs
13. Anticancer Drugs (Antineoplastic Drugs)..........................................................................................................................169
14. Miscellaneous Drugs ..............................................................................................................................................................176
Immunosuppressant Drugs, Chelating Agents, Locally Acting Drugs on Skin and Mucous Membranes, Drugs for Acne
vulgaris, Antiseptics and Disinfectants, Ectoparasiticides, Vaccines, Antisera and Immune Globulins
Index of Nonproprietary Names of Drugs..................................................................................................................................195
Index of Proprietary (Brand) Names of Drugs ..........................................................................................................................211
DrugsActing onAutonomic Nervous System
1
3
Anticholinergic Drugs
Drugs Acting on Autonomic Nervous System
6
Adrenergic Drugs 7
10 Drugs Acting on Autonomic Nervous System
12 Drugs Acting on Autonomic Nervous System
14 Drugs Acting on Autonomic Nervous System
Autacoids and Related Drugs
2
19
Drugs for Migraine
21
Prostaglandins (PGs)
23
Nonsteroidal Antiinflammatory Drugs/ Antipyretic-Analgesics
27
Antirheumatoid Drugs/Drugs for Gout
Drugs for Respiratory Disorders
3
Drugs for Bronchial Asthma 33
Hormones and Related Drugs
4
Thyroid Hormone and Thyroid Inhibitors 39
Hormones and Related Drugs
40
Hormones and Related Drugs
42
Hormones and Related Drugs
44
Androgens and Related Drugs 47
Hormones and Related Drugs
50
53
Progestins
55
Hormonal Contraceptives
Hormones and Related Drugs
58
DrugsActing on Peripheral (somatic) Nervous System
5
Drugs Acting on Peripheral (somatic) Nervous System
62
DrugsActing on Central Nervous System
6
Drugs Acting on Central Nervous System
66
Sedative-Hypnotic Drugs 67
Antiepileptic Drugs 69
Drugs Acting on Central Nervous System
72
Antipsychotic Drugs 75
77
Drugs for Mania and Bipolar Disorder
79
Antidepressants
Opioid Analgesics and Antagonists 83
CNS Stimulants and Cognition Enhancers 85
Cardiovascular Drugs
7
Antihypertensive Drugs 89
Antianginal Drugs 93
Drugs for Peripheral Vascular Diseases 95
Drugs for Congestive Heart Failure 97
Antiarrhythmic Drugs 99
DrugsActing on Kidney
8
DrugsAffecting Blood
9
Coagulants 109
Anticoagulants 111
Drugs Affecting Blood
116
Gastrointestinal Drugs
10
Gastrointestinal Drugs
122
Laxatives 125
Gastrointestinal Drugs
128
130
Antibacterial Drugs
11
Sulfonamides/Quinolone Antimicrobials 131
Antibacterial Drugs
134
Cephalosporins 137
Antitubercular Drugs 145
Antitubercular/Antileprotic Drugs 147
Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs
12
Antiviral Drugs (Non-retroviral) 153
Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs
154
Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs
158
Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs
162
Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs
166
Anticancer Drugs (Antineoplastic Drugs)
13
Anticancer Drugs (Antineoplastic Drugs)
170
171
Anticancer Drugs
176
Miscellaneous Drugs
14
Miscellaneous Drugs
184
ANTISEPTICS AND DISINFECTANTS
1. Phenol derivatives:
Phenol, Cresol, Hexylresorcinol, Chloroxylenol, Hexachlorophene.
2. Oxidizing agents:
Pot. permangnate, Hydrogen peroxide, Benzoyl peroxide.
3. Halogens:
Iodine, Iodophores, Chlorine, Chlorophores.
4. Biguanide
Chlorhexidine.
5. Quaternary ammonium (Cationic);
Cetrimide, Benzalkonium chloride (Zephiran), Dequalinium chloride.
6. Soaps
of Sod. and Pot.
7. Alcohols
Ethanol, Isopropanol.
8. Aldehydes
Formaldehyde, Glutaraldehyde.
Miscellaneous Drugs
186
9. Acids
Boric acid, Acetic acid.
10. Metallic salts
Silver nitrate, Silver sulfadiazine, Mild silver protein, Zinc sulfate, Calamine, Zinc oxide.
11. Dyes
Gentian violet, Brilliant green, Acriflavine, Proflavine.
12. Furan derivative
Nitrofurazone.
Vaccines 189
Miscellaneous Drugs
192
Antisera (from Horse)
Tetanus antitoxin (ATS)
Gas gangrene antitoxin (AGS)
Diphtheria antitoxin (ADS)
Antirabies serum (ARS)
Antisnake venom polyvalent
Immune globulins (Human)
Normal human gamma globulin
Rho(D) immune globulin
Tetanus immune globulin
Rabies immune globulin
Hepatitis-B immune globulin

KD Tripathi Classification of Drugs.pptx

  • 1.
    Pharmacological CLASSIFICATION OF DRUGS withDoses and Preparations FIFTH EDITION KD Tripathi MD Ex-Director-Professor and Head of Pharmacology Maulana Azad Medical College and associated LN and GB Pant Hospitals, New Delhi JAYPEE BROTHERS MEDICAL PUBLISHERS (P) LTD New Delhi • London • Philadelphia • Panama ®
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    1. Drugs Actingon Autonomic Nervous System .....................................................................................................................1 Cholinergic Drugs, Anticholinergic Drugs, Ganglionic Stimulants, Ganglionic Blocking Agents, Adrenergic Drugs, -Adrenergic Blocking Drugs, -Adrenergic Blocking Drugs, Topical Drugs for Glaucoma 2. Autacoids and Related Drugs.................................................................................................................................................16 Histaminergic Agonists, H1-Antagonists, 5-Hydroxytryptamine (5-HT) Antagonists, Drugs for Migraine, Prostaglandins (PGs), Nonsteroidal Antiinflammatory Drugs (NSAIDs)/Antipyretic Analgesics, Antirheumatoid Drugs, Drugs for Gout 3. Drugs for Respiratory Disorders............................................................................................................................................29 Drugs for Cough, Drugs for Bronchial Asthma 4. Hormones and Related Drugs ................................................................................................................................................37 Anterior Pituitary Hormones, Drugs Altering Anterior Pituitary Hormone Secretion, Thyroid Hormone, Thyroid Inhibitors, Insulins, Oral Antidiabetic Drugs, Corticosteroids, Topical Steroids, Androgens and Related Drugs, Drugs for Erectile Dysfunction, Estrogens and Related Drugs, Progestins, Hormonal Contraceptives, Uterine Stimulants, Uterine Relaxants 5. Drugs Acting on Peripheral (somatic) Nervous System...................................................................................................60 Skeletal Muscle Relaxants, Local Anaesthetics 6. Drugs Acting on Central Nervous System ..........................................................................................................................64 General Anaesthetics, Preanaesthetic Medication Drugs, Sedative-Hypnotic Drugs, Antiepileptic Drugs, Antiparkinsonian Drugs, Antipsychotic Drugs, Drugs for Mania and Bipolar Disorder, Hallucinogens, Antidepressants, Antianxiety Drugs, Opioid Analgesics and Antagonists, Central Nervous System (CNS) Stimulants, Cognition Enhancers 7. Cardiovascular Drugs ...............................................................................................................................................................88 Antihypertensive Drugs, Antianginal Drugs, Drugs for Peripheral Vascular Diseases, Drugs for Congestive Heart Failure, Antiarrhythmic Drugs Contents
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    Pharmacological Classification ofDrugs with Doses and Preparations xii 8. Drugs Acting on Kidney........................................................................................................................................................102 Diuretics, Antidiuretics 9. Drugs Affecting Blood ...........................................................................................................................................................105 Haematinics, Coagulants, Anticoagulants, Fibrinolytics, Antifibrinolytics, Antiplatelet Drugs, Hypolipidaemic Drugs, Plasma Expanders 10. Gastrointestinal Drugs ...........................................................................................................................................................118 Drugs for Peptic Ulcer, Antiemetics, Laxatives, Drugs for Diarrhoea 11. Antibacterial Drugs.................................................................................................................................................................130 Antibacterial Drugs, Sulfonamides, Quinolone Antimicrobials, Penicillins, Cephalosporins, Monobactams, Carbapenems, Aminoglycoside Antibiotics, Tetracyclines, Chloramphenicol, Macrolide Antibiotics, Lincosamide Antibiotics, Aminocyclitol Antibiotic, Glycopeptide Antibiotics, Oxazolidinone, Polypeptide Antibiotics, Urinary Antiseptics, Antitubercular Drugs, Antileprotic Drugs 12. Antifungal, Antiviral, Antiprotozoal and Anthelmintic Drugs....................................................................................150 Antifungal Drugs, Antiviral Drugs (Non-retroviral), Antiretrovirus Drugs, Antimalarial Drugs, Antiamoebic Drugs, Drugs for Giardiasis, Drugs for Trichomoniasis, Drugs for Leishmaniasis, Anthelmintic Drugs 13. Anticancer Drugs (Antineoplastic Drugs)..........................................................................................................................169 14. Miscellaneous Drugs ..............................................................................................................................................................176 Immunosuppressant Drugs, Chelating Agents, Locally Acting Drugs on Skin and Mucous Membranes, Drugs for Acne vulgaris, Antiseptics and Disinfectants, Ectoparasiticides, Vaccines, Antisera and Immune Globulins Index of Nonproprietary Names of Drugs..................................................................................................................................195 Index of Proprietary (Brand) Names of Drugs ..........................................................................................................................211
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    Drugs Acting onAutonomic Nervous System 6
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    10 Drugs Actingon Autonomic Nervous System
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    12 Drugs Actingon Autonomic Nervous System
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    14 Drugs Actingon Autonomic Nervous System
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    Thyroid Hormone andThyroid Inhibitors 39
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    DrugsActing on Peripheral(somatic) Nervous System 5
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    Drugs Acting onPeripheral (somatic) Nervous System 62
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    DrugsActing on CentralNervous System 6
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    Drugs Acting onCentral Nervous System 66
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    Drugs Acting onCentral Nervous System 72
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    77 Drugs for Maniaand Bipolar Disorder
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    Opioid Analgesics andAntagonists 83
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    CNS Stimulants andCognition Enhancers 85
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    Drugs for PeripheralVascular Diseases 95
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    Drugs for CongestiveHeart Failure 97
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    Antifungal, Antiviral, Antiprotozoaland Anthelmintic Drugs 12
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    Antifungal, Antiviral, Antiprotozoaland Anthelmintic Drugs 154
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    Antifungal, Antiviral, Antiprotozoaland Anthelmintic Drugs 158
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    Antifungal, Antiviral, Antiprotozoaland Anthelmintic Drugs 162
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    Antifungal, Antiviral, Antiprotozoaland Anthelmintic Drugs 166
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    ANTISEPTICS AND DISINFECTANTS 1.Phenol derivatives: Phenol, Cresol, Hexylresorcinol, Chloroxylenol, Hexachlorophene. 2. Oxidizing agents: Pot. permangnate, Hydrogen peroxide, Benzoyl peroxide. 3. Halogens: Iodine, Iodophores, Chlorine, Chlorophores. 4. Biguanide Chlorhexidine. 5. Quaternary ammonium (Cationic); Cetrimide, Benzalkonium chloride (Zephiran), Dequalinium chloride. 6. Soaps of Sod. and Pot. 7. Alcohols Ethanol, Isopropanol. 8. Aldehydes Formaldehyde, Glutaraldehyde.
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    Miscellaneous Drugs 186 9. Acids Boricacid, Acetic acid. 10. Metallic salts Silver nitrate, Silver sulfadiazine, Mild silver protein, Zinc sulfate, Calamine, Zinc oxide. 11. Dyes Gentian violet, Brilliant green, Acriflavine, Proflavine. 12. Furan derivative Nitrofurazone.
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    Miscellaneous Drugs 192 Antisera (fromHorse) Tetanus antitoxin (ATS) Gas gangrene antitoxin (AGS) Diphtheria antitoxin (ADS) Antirabies serum (ARS) Antisnake venom polyvalent Immune globulins (Human) Normal human gamma globulin Rho(D) immune globulin Tetanus immune globulin Rabies immune globulin Hepatitis-B immune globulin