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Neuromuscular blocking agents
1. PHARMACOLOGY-I
Session 2020-21
Submitted by –
Mr. Suyash Jain
Department Of Pharmaceutical Sciences
Dr. Harisingh Gour Vishwavidyalaya, Sagar (M.P.)
Neuromuscular blocking agents
( A Central University )
8. NEUROMUSCULAR
STIMULATORS
Drugs having acetylcholine like action-
Methacholine,Carbachol& Nicotin
But these are either not destroyed or destroyedvery
slowly by acetylcholinesterase so causes repeated
stimulation & continuous action of muscle –Muscle
spasm.
9. NEUROMUSCULAR
STIMULATORS
Drugs that Inactivatethe enzyme Cholinesterase
(Anticholinesterase)–Neostigmine,
Physostigmine&Disopropylflurophosphate
(DFP)
So it leads to repeated stimulation & continuous action of
muscle. E.g–Laryngeal Spasm.