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Reseptor Adenergik
 Reseptor adrenergik adalah glikoprotein cell surface yang
mengenali dan secara selektif mengikat katekolamin,
norepinefrin dan epinefrin, yang dilepaskan dari ujung
saraf simpatik dan medula adrenal
 Reseptor adrenergik dibagi pada dua kategori umum: α
dan β
 Kemdian dibagi menjadi dua subtipe: α1 dan α2, β1 dan β2
dan β3
• Target Respon Reseptor Adrenergik:
• Reseptor α adrenergik,
Alpha-1: kontraksi vascular dan otot polos genitourinary.
Alpha-2: kontraksi vacular smooth muscle, inhibisi pelepasan
insulin, induksi pelepasan glukagon, agregasi platelet dan inhibisi
presinaptik dari norepinefrin
• Reseptor β adrenergik
Beta-1 : positif inotropic dan chronotropic efek pada jantung
menaikkan heart rate (jumlah denyut jantung perunit waktu),
menaikkan kontraksi jantung
Beta-2: relaksasi vaskular, bronkial, gastrointestinal dan otot polos
genitourinary; menstimulasi glyconenolysis dan gluconeogenesis di
hati.
Beta-3: lipolisis di jaringan adiposa
Degradasi Katekolamin
Perkembangan hormon katekolamin
 Sympathetic hyperactivity

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up1.pptx

  • 1. Reseptor Adenergik  Reseptor adrenergik adalah glikoprotein cell surface yang mengenali dan secara selektif mengikat katekolamin, norepinefrin dan epinefrin, yang dilepaskan dari ujung saraf simpatik dan medula adrenal  Reseptor adrenergik dibagi pada dua kategori umum: α dan β  Kemdian dibagi menjadi dua subtipe: α1 dan α2, β1 dan β2 dan β3
  • 2. • Target Respon Reseptor Adrenergik: • Reseptor α adrenergik, Alpha-1: kontraksi vascular dan otot polos genitourinary. Alpha-2: kontraksi vacular smooth muscle, inhibisi pelepasan insulin, induksi pelepasan glukagon, agregasi platelet dan inhibisi presinaptik dari norepinefrin • Reseptor β adrenergik Beta-1 : positif inotropic dan chronotropic efek pada jantung menaikkan heart rate (jumlah denyut jantung perunit waktu), menaikkan kontraksi jantung Beta-2: relaksasi vaskular, bronkial, gastrointestinal dan otot polos genitourinary; menstimulasi glyconenolysis dan gluconeogenesis di hati. Beta-3: lipolisis di jaringan adiposa
  • 4. Perkembangan hormon katekolamin  Sympathetic hyperactivity