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CETRIZINE
BY:- ATIF KHAN
BSC BT II YEAR
MECHANISM OF
ACTION
Cetirizine competes with histamine for
binding at H1-receptor sites on the
effector cell surface, resulting in
suppression of histaminic edema, flare,
and pruritus.
Cetirizine is a non-sedating antihistamine
that works by blocking histamine (H-1)
receptors on cells.
 It is similar to the other second
generation antihistamines
DESCRIPTION
A potent second-generation histamine
H1 antagonist that is effective in the
treatment of allergic rhinitis, chronic
urticaria, and pollen-induced asthma.
Unlike many traditional antihistamines,
it does not cause drowsiness or
anticholinergic side effects.
Cetirizine and other second-generation
antihistamines do not readily enter the
brain from the blood, and, therefore,
they cause less drowsiness.
Used to relieve allergy symptoms
such as
 watery eyes
 runny nose
 itching eyes/nose
 sneezing
Common side effects include
 headache
 dry mouth
 feeling sick
 dizziness
 tummy pain
 diarrhoea.
THANK YOU

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Cetrizine

  • 2.
  • 3. MECHANISM OF ACTION Cetirizine competes with histamine for binding at H1-receptor sites on the effector cell surface, resulting in suppression of histaminic edema, flare, and pruritus. Cetirizine is a non-sedating antihistamine that works by blocking histamine (H-1) receptors on cells.  It is similar to the other second generation antihistamines
  • 4. DESCRIPTION A potent second-generation histamine H1 antagonist that is effective in the treatment of allergic rhinitis, chronic urticaria, and pollen-induced asthma. Unlike many traditional antihistamines, it does not cause drowsiness or anticholinergic side effects. Cetirizine and other second-generation antihistamines do not readily enter the brain from the blood, and, therefore, they cause less drowsiness.
  • 5. Used to relieve allergy symptoms such as  watery eyes  runny nose  itching eyes/nose  sneezing
  • 6. Common side effects include  headache  dry mouth  feeling sick  dizziness  tummy pain  diarrhoea.