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FARMAKOLOGI
Nurma Suri, M. Biomed.Sc. MKM., Apt
UNIVERSITAS MUHAMMADIYAH PRINGSEWU
PROGRAM STUDI DIII KEPERAWATAN
TAHUN 2020
MATERI BAHAN AJAR
APA ITU FARMAKOLOGI
ISTILAH –ISTILAH FARMAKOLOGI
FARMAKOKINETIKA
FARMAKODINAMIKA
KLASIFIKASI PENGGOLONGAN OBAT
OBAT SSP DAN OTONOM
ANASTESI
NSAID
DIURESIS
HEMATOLOGI NURMA SURI, M. BIOMED, Sc, MKM,APT
KONSEP FARMAKOLOGI
Nurma Suri, M. Biomed.Sc. MKM., Apt
UNIVERSITAS MUHAMMADIYAH PRINGSEWU
PROGRAM STUDI DIII KEPERAWATAN
TAHUN 2020
FARMASETIKA
FARMAKOLOGI
FARMAKOTERAPI
FARMAKOKINETIK
FARMAKODINAMIK
EFEK POSITIF/NEGATIF
TERAPI OBAT KEPADA
PASIEN
MEPRODUKSI OBAT
DALAM BENTUK SEDIAAN
YANG TEPAT BAGI PASIEN
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
OBAT
DIKONSUMSI
OBAT
MEMBERIKAN
EFEK TERAPI
?
O
B
A
T
FARMAKOLOGI  ILMU MENGENAI
PENGARUH SENYAWA TERHADAP SEL
HIDUP MELALUI PROSES KIMIA
NURMA SURI, M. BIOMED, Sc, MKM,APT
URINE
FESES
KERINGAT
DARAH
MEMBRAN SEL
OBAT PROTEIN
OBAT
BEBAS
OBAT
BEBAS
RESEPTOR
FARMAKOKINETIK
FARMAKODINAMIK
2/28/2020
NURMA SURI, M. BIOMED, Sc, MKM,APT
2/28/2020
FARMAKOKINETIK
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
OBAT + RESEPTOR OBAT-RESEPTOR EFEK TERAPI
ACE INHIBITOR
B-BLOKER ADRENALIN
DNA
VOLTAGE GATED IONCHANEL
ENZIM-LINKED RESEPTOR
FARMAKODINAMIK
2/28/2020
NURMA SURI, M. BIOMED, Sc, MKM,APT
KETERSEDIAAN HAYATI =
FRAKSI DARI DOSIS OBAT
DIBERIKAN YANG DAPAT
MENCAPAI SIRKULASI SISTEMIK
TINGKAT DI MANA OBAT
AKTIF DIKELUARKAN DARI
TUBUH
UKURAN
KEMAMPUAN OBAT UNTUK
BERIKATAN PADA RESEPTOR2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
APA YANG TERJADI PADA OBAT SAAT
DIBERIKAN KEPADA MAKHLUK HIDUP
TUBUH  OBAT
FARMAKOKINETIK FARMAKODINAMIK
APA YANG TERJADI PADA MAKHLUK
HIDUP SAAT DIBERIKAN OBAT
OBAT  TUBUH
DOSIS TERAPI
DOSIS TOKSIK
SUB-DOSIS
THERAUPHETIC
WINDOW
ONSET OF
EFFECT
MENGAPA CARA MINUM OBAT
BERBEDA-BEDA?
1 X 1 TABLET
2 X 1 TABLET
3 X 1 TABLET
MENGAPA ANTIBIOTIK HARUS
DIMINUM TEPAT WAKTU?
CARI
DEFINISI
DIBUKU
TUGAS
BAGAIMANA
GRAFIK
FARMAKOKINETIK
UNTUK OBAT
YANG DIBERIKAN
SECARA
INTRAVENA (IV)
DAN OBAT
TOPIKAL (SALEP)
2/28/2020
NURMA SURI, M. BIOMED, Sc, MKM,APT
SEL JARINGAN ORGAN
SISTEM
ORGAN
NURMA SURI, M. BIOMED, Sc, MKM,APT
ATC = THE ANATOMICAL THERAUPETIC CHEMICAL
SISTEM KLASIFIKASI OBAT YANG MENGKLASIFIKASIKAN BAHAN AKTIF
OBAT SESUAI DENGAN ORGAN ATAU SISTEM DI MANA OBAT BEKERJA,
EFEK TERAPI OBAT, FARMAKOLOGI DAN KANDUNGAN KIMIA.
OBAT SISTEM
SARAF
SARAF PUSAT
SARAF OTONOM
ANASTESI
NYERI
OBAT
DIURETIK
OBAT
KARDIOVASKULAR
HEMATOLOGI
OBAT HORMON
OBAT SISTEM
PENCERNAAN
WHO
OBAT
REPRODUKSI
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
FARMAKOKINETIK
Nurma Suri, M. Biomed.Sc. MKM., Apt
UNIVERSITAS MUHAMMADIYAH PRINGSEWU
PROGRAM STUDI DIII KEPERAWATAN
TAHUN 2020
FARMAKOKINETIK
APA YANG TERJADI PADA OBAT SAAT DIBERIKAN
KEPADA MAKHLUK HIDUP A-D-M-E
TUBUH  OBAT
A
DM
E
bsorbsi
istribusietabolisme
kskresi
PROSES MASUKNYA OBAT
DARI TEMPAT PEMBERIAN KE
DALAM DARAH
PROSES PENYEBARAN OBAT
MELALUI DARAH KE SELURUH
JARINGAN TUBUH
PROSES PERUBAHAN ATAU
MODIFIKASI OBAT DIDALAM
TUBUH
PROSES PENGELUARAN OBAT
DARI DALAM TUBUH
NURMA SURI, M. BIOMED, Sc, MKM,APT
FARMAKOKINETIK A bsorbsi
BENTUK SEDIAAN
OBAT
USUS  PANJANG 280 CM,
DIAMETER 4 CM, DISERTAI
VILI DAN MIKROVILI
SUBLINGUAL 
LUAS
PERMUKAAN
ABSORBSI
KECIL.
LANGSUNG KE
VENA KAVA
SUPERIOR
50% DARAH
DARI REKTUM
MELALUI
VENA PORTA
NURMA SURI, M. BIOMED, Sc, MKM,APT
DIFUSI PASIFENDOSITOSIS
TRANSPORT
MEMBRAN
INTRASELULAR
MEKANISME
ABSORBSI OBAT
INTERAKSI
• OBAT-OBAT
• OBAT-MAKANAN
ATURAN PAKAI
OBAT !!!
MEMBRAN
PLASMA
LIPOFILIK
NURMA SURI, M. BIOMED, Sc, MKM,APT
FARMAKOKINETIK D istribusi
KOMPOSISI DARAH
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
1. ALBUMIN : MENGIKAT
OBAT-OBAT ASAM DAN
OBAT-OBAT NETRAL
2. ALPHA GLIKOPROTEIN :
MENGIKAT OBAT-OBAT
BASA
3. KORTIKOSTEROID BINDING
GLOBULIN (CBG):
MENGIKAT
KORTIKOSTEROID
4. SEX STEROID BINDING
GLOBULIN (SSBG)
MENGIKAT HORMON
KELAMIN
MACAM PROTEIN
PLASMA
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
FARMAKOKINETIK M etabolisme
OBAT LARUT LEMAK
OBAT LARUT AIR
EKSKRESI
REAKSI FASE I
(PENAMBAHAN GUGUS
POLAR)
• OKSIDASI
• REDUKSI
• HIDROLISIS
REAKSI FASE II
• KONJUGASI DENGAN
SUBSTRAT ENDOGEN
(AS.GLUKORONAT,
AS.SULFAT, AS.
ASETAT, AS. AMINO)
HATI, DINDING USUS, GINJAL,
PARU, DARAH, OTAK, KULIT
NURMA SURI, M. BIOMED, Sc, MKM,APT
FARMAKOKINETIK E kskresi
FUNGSI GINJAL
MENGALAMI
KEMATANGAN
USIA 6-12 BULAN,
SETELAH DEWASA
MENURUN 1%
PER TAAHUN
GFR (GLOMERULAR FILTRATION RATE)
ATAU LFG (LAJU FILTRASI GLOMERULUS) 
KELUARAN KREATININ (CREATININE CLEARANCE
IBU MEYUSUI
pH !!!
FARMAKODINAMIK
Nurma Suri, M. Biomed.Sc. MKM., Apt
UNIVERSITAS MUHAMMADIYAH PRINGSEWU
PROGRAM STUDI DIII KEPERAWATAN
TAHUN 2020
• RESEPTOR
• ENZYM
• TRANSPORTER
• ION CHANEL
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
INTERAKSI OBAT DAN RESEPTOR
SPESIFISITAS
SELEKTIVITAS
KERJA OBAT TERBATAS PADA SATU JENIS RESEPTOR
KERJA OBAT PADA DOSIS RENDAH HANYA
MENGHASILKAN SATU EFEK
AGONIS
ANTAGONIS
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
SPESIFISITAS
SELEKTIVITAS
DOSIS TERAPI
DOSIS TOKSIK
SUB-DOSIS
THERAUPHETIC
WINDOW
ONSET OF
EFFECT
MENGAPA CARA MINUM OBAT
BERBEDA-BEDA?
1 X 1 TABLET
2 X 1 TABLET
3 X 1 TABLET
MENGAPA ANTIBIOTIK HARUS
DIMINUM TEPAT WAKTU?
CARI
DEFINISI
DIBUKU
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
TUGAS
CARI SATU
JENIS OBAT
YANG
BEKERJA
PADA SISTEM
SARAF PUSAT
ATAU SISTEM
SARAF
OTONOM
VIDEO
MEKANISME
KERJA OBAT
PELAJARI
DISKUSI, PRESENTASI,
DAN QUIZ
Nurma Suri, M. Biomed.Sc. MKM., Apt
UNIVERSITAS MUHAMMADIYAH PRINGSEWU
PROGRAM STUDI DIII KEPERAWATAN
TAHUN 2020
MAHASISWA MAMPU MENJELASKAN KONSEP FARMAKOLOGI
YANG TERDIRI DARI FARMAKOKINETIK DAN FARMAKODINAMIK
MENGGUNAKAN
GAMBAR DISAMPING
JELASKAN KONSEP
FARMAKOLOGI,
FARMAKOKINETIK
DAN
FARMAKODINAMIK
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
MAHASISWA MAMPU MENJELASKAN KONSEP FARMAKOLOGI
YANG TERDIRI DARI FARMAKOKINETIK DAN FARMAKODINAMIK
MENGGUNAKAN
GAMBAR DISAMPING
JELASKAN KONSEP
FARMAKODINAMIK
DAN BERIKAN
CONTOHNYA
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
MAHASISWA MAMPU MENJELASKAN KONSEP FARMAKOLOGI
YANG TERDIRI DARI FARMAKOKINETIK DAN FARMAKODINAMIK
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
MAHASISWA MAMPU MENJELASKAN KONSEP FARMAKOLOGI
YANG TERDIRI DARI FARMAKOKINETIK DAN FARMAKODINAMIK
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
MAHASISWA MAMPU MENGKAITKAN KONSEP FARMAKOLOGI
PADA APLIKASINYA DI DUNIA KEPERAWATAN
POINT-POINT
YANG PERLU
DIPERHATIKAN
DALAM
KEPERAWATAN
KAITANNYA
DENGAN ILMU
FARMAKOLOGI
2/28/2020 NURMA SURI, M. BIOMED, Sc, MKM,APT
TERIMA KASIH
STUDY HARD
PLAY HARD
PRAY HARD

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