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Bromocriptine Trade name: parlodel Class: Antiparkinson agent
Dosage form available ,[object Object],[object Object]
Pharmacology   ,[object Object]
Pharmacokinetic data   1-2 h   Onset   Major elimination route is hepatic; 6% is renally eliminated .  Terminal half - life of 15 h  Elimination   Primarily metabolized in the GI tract and liver  ( CYP3A4 ).  Undergoes extensive first - pass metabolism   Metabolism   to 96% bound to serum albumin   90   Distribution   of oral dose absorbed   28% Absorption
Indications and Usage ,[object Object],[object Object],[object Object],[object Object]
Dose ,[object Object],[object Object],[object Object]
[object Object],[object Object],[object Object]
Contraindications   ,[object Object],[object Object],[object Object]
Adverse Reactions ,[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
[object Object],[object Object],[object Object],[object Object],[object Object],[object Object]
Drugs ineraction ,[object Object],[object Object]
[object Object],[object Object],[object Object],[object Object],[object Object]
[object Object],[object Object],[object Object],[object Object],[object Object]
General Advice ,[object Object],[object Object]

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Bromocriptine

  • 1. Bromocriptine Trade name: parlodel Class: Antiparkinson agent
  • 2.
  • 3.
  • 4. Pharmacokinetic data 1-2 h Onset Major elimination route is hepatic; 6% is renally eliminated . Terminal half - life of 15 h Elimination Primarily metabolized in the GI tract and liver ( CYP3A4 ). Undergoes extensive first - pass metabolism Metabolism to 96% bound to serum albumin 90 Distribution of oral dose absorbed 28% Absorption
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