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Promising New
Cancer Drugs
(Jan 2024)
Source: FDA
Molecule Brand Name Manufacturer
Name Phase (Jan 2024)
ATR inhibitor + PDL-1 mAb
PD-1/CTLA-4
bispecific mAb Volrustomig
STING Agonist TAK-500
Ceralasertib + Imfinzi Phase III, expected filing in 2024
Phase III, new to this phase
Phase III
Phase II
BTK inhibitor + R-CHOP Calquence + R-CHOP
Phase II
Phase II
Source: FDA
Molecule Brand Name Manufacturer
Name Phase (Jan 2024)
CD27 agonist mAb
BTK inhibitor + BCL-2
inhibitor + anti-CD20 mAb
Calquence + venetoclax +
obinutuzumab
Targeted Next Generation
Interferon
EGFR x CD3 Conditional T-
cell engager
Modakafusp Alfa
TAK-186
Boserolimab
Phase II, in combination with KEYTRUDA
Phase II
Phase II
Source: FDA
Molecule Brand Name Manufacturer
Name Phase (Jan 2024)
SUMOylation Inhibitor
Anaplastic Lymphoma
Kinase (ALK) inhibitor Brigatinib
EGFR/HER2 inhibitor mobocertinib
Subasumstat (TAK-981)
Phase II
Phase II

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Promising New Cancer Drugs Jan 2024 by Insights10

  • 2. Source: FDA Molecule Brand Name Manufacturer Name Phase (Jan 2024) ATR inhibitor + PDL-1 mAb PD-1/CTLA-4 bispecific mAb Volrustomig STING Agonist TAK-500 Ceralasertib + Imfinzi Phase III, expected filing in 2024 Phase III, new to this phase Phase III Phase II BTK inhibitor + R-CHOP Calquence + R-CHOP
  • 3. Phase II Phase II Source: FDA Molecule Brand Name Manufacturer Name Phase (Jan 2024) CD27 agonist mAb BTK inhibitor + BCL-2 inhibitor + anti-CD20 mAb Calquence + venetoclax + obinutuzumab Targeted Next Generation Interferon EGFR x CD3 Conditional T- cell engager Modakafusp Alfa TAK-186 Boserolimab Phase II, in combination with KEYTRUDA Phase II
  • 4. Phase II Source: FDA Molecule Brand Name Manufacturer Name Phase (Jan 2024) SUMOylation Inhibitor Anaplastic Lymphoma Kinase (ALK) inhibitor Brigatinib EGFR/HER2 inhibitor mobocertinib Subasumstat (TAK-981) Phase II Phase II