LIST OF THE INTERMEDIATES
- 1. LIST OF THE INTERMEDIATES:
I TRITYL OLMESARTAN
II CLOPIDOGREL BISULPHATE
01 S-(+)-2-chlorophenylglycinemethyl ester
[141109- 14-4]
02 S-(+)-Methyl-(2-chlorophenyl)[(2-(2-thienyl)amino] acetate hydrochloride (OR) (+) - 2 -
(2-Chlorophenyl)-N- [2-(2-thienyl)ethyl]glycine methyl esterhydrchloride
[141109- 20-8]
03 4,5,6,7 – TetrahydroThieno(3,2-c) PyridineHCl
04 ClopidogrelCamphorSulfonate (CPCSA SALT)
III LOSARTAN POTASSIUM
01 2-Cyano-4’-bromomethylbiphenyl
[114772-54-2]
02 Trityl Losartan
[133909-99-6]
03 2-Butyl -4-chloro-[(2'-cyanobiphenyl-4-yl)-methyl ]-5-(hydroxymethyl)imidazole
[114772-55-3]
03 (1-((2'-(2H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazol-5-
yl)methanol(OR) Losartan
[114798-26-4]
IV EMTRICITABINE
01 (2R,SR)-5-Hydroxy-[1,3]-oxathiolane-2-carboxylicacid,ester2S-isopropyl–5R – methyl
-1R – Cyclohexylester
[147126-62-3]
02 (1R, 2S,SR) – Methyl – (2R, SS) – 5-[4-amino-5-fuoro-2-oxo-
2H – pyrinidin-1-yl](1,2) oxathiolane-2-carboxylicacid(FCE)
[147126-75-8]
- 2. VII PANTOPRAZOLE SODIUM
01 5-(Difluoromethoxy)-2[[(3,4-dimethoxy-2-pyridinyl)methyl]thio]-1H-benzimidazole
[102625-64-9]
02 5-(Difluoromethoxy)-2[[(3,4-dimethoxy-2-pyridinyl)methyl]sulfinyl]-1H-benzimidazole
(OR) Pantoprazole [142678-34-0]
VIII SERTRALINE HYDROCHLORIDE
01 4-(3,4-Dichlorophenyl)-3,4-dihyro-1-(2H)-naphthalenone [75560-19-3]
IX CETIRIZINE DIHYDROCHLORIDE
01 1-(4-Chlrodiphenylmethyl)-piperazine [303-26-4]
02 4-Chlorobenzhydrylchloride [134-83-8]
X FLUCONAZOLE/ VORICONAZOLE
01 2,4-difluoro-2-(1H-1,2,4-triazole-1yl)acetophenone (OR) 1-(2,4-Difluorophenyl)-2-(1H-
1,2,4-Triazole-1-yl) Ethanone [86404-63-9]
02 [2(2,4-difluorophenyl)-1-(1H-1,2,4-triazole-1-yl)2,3epoxypropane methane sulphonate
XI PREGABALIN
01 2-Carboxyethyl-3-cyano-5-methylhexanoicacidethyl ester
02 3-Aminomethyl-5-methyl haxanoicacid(racemicPregabalin)
03 3-Carbamoylmethyl-5-methyl-hexanoicacid
XII LEVOCETIRIZINE DIHYDROCHLORIDE
01 (-) 1-(4-Chlorophenyl)phenylmethyl amine
02 (-)-1-(4-chlorophenylmethyl)-piperazine
XIII TELMISARTAN
01 Methyl 4-(bromomethyl)-2-biphenyl-2-carboxylate
XIV VALSARTAN
N – [(2-eqanobiphenyl-4-yl)methyl] –(L) – valine methylesterhydrochloride