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Reflecting the dose and half life - on pharma minutes is
leading the minute ‘s response element
Formulating the minute application produce knowledge
and reflect receptor site class .
The drug has a
ngligible effects at
alpha and
muscarinic recptors.
t1/2 about
10minutes
patient
Metoprolol (Lopressor,Toprol) , Atenolol (Tenormin)
Metoprolol (Lopressor,Toprol) , Atenolol (Tenormin)
Since their B1 selectivity is rather modest ,they should be used with great caution , if at all in patients with
history of bronchospasm .
They are effective in the major cardiovascular applications of beta – blocking group (hypertension and
angina).
patients with history
of bronchospasm
Metoprolol (Lopressor,Toprol) , Atenolol (Tenormin)
And
other drugs
are members of B1 selective group
Metoprolol (Lopressor,Toprol) , Atenolol (Tenormin)
Metoprolol & Atenolol
These agents may be safer in patients who
experience bronchoconstrictuve responses
to propranolol .
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